A

Abdollahi-Roodsaz, Shahla, van de Loo, Fons, Koenders, Marije, Helsen, Monique, Walgreen, Brigitte, van den Bersselaar, Leduine, Arntz, Onno, Takahashi, Nozomi, Joosten, Leo and van den Berg, Wim (2011) Destructive Role of Myeloid Differentiation Factor 88 and Protective Role of TIR-Containing Adaptor Inducing Interferon β in IL-17-Dependent Arthritis. Arthritis & Rheumatism. ISSN 0004-3591

Abraham, Jinu, Prajapati, Suresh, Nishijo, Koichi, Schaffer, Beverly S, Taniguchi, Eri, Kilcoyne, Aoife, McCleish, Amanda T, Zarzabal, Lee Ann, Michalek, Joel E, Nelon, Laura D, Giles, Francis G, Efstratiadis, Argiris, LeGallo, Robin D, Nowak, Brent M, Rubin, Brian P, Keller, Charles and Jeay, Sebastien (2011) Evasion mechanisms to Igf1r inhibition in rhabdomyosarcoma. Molecular Cancer Therapeutics, 10 (4). pp. 697-707. ISSN 1535-7163

Agarwal, Abhiruchi, Boettcher, Andreas, Kneuer, Rainer, Sari-Sarraf, Farid, Donovan, Adriana, Woelcke, Julian and Krucker, Thomas (2011) Quantitative and functional assessment of treatment strategies for acute pancreatitis with optical fluorescence imaging in rats. Plos, 8 (2). e55959. ISSN 1932-6203

Allyson, Julie, Dontigny, Eve, Cyr, Michel, Massicotte, Guy and Auberson, Yves (2011) Blockade of NR2A-containing NMDA Receptors Induces Tau Phosphorylation in Rat Hippocampal Slices. Neural Plasticity. p. 340168. ISSN 0792-8483

Anders, Lars, Ke, Nan, Hydbring, Per, Zhai, Huili, Choi, Yoon, Braun, Pascal, Vidal, Marc and Sicinski, Peter (2011) a systematic substrate screen links CDK4/6 to senescence suppression through FOXM1. Cancer Cell, 20 (5). pp. 620-634. ISSN 1535-6108

Anemona, Alessandra, Basile, Venere, Hilbert, Anne-Katrin, Rondini, Simona, Micoli, Francesca, Marchetti, Elisa, Di Cioccio, Vito, Saul, Allan, Martin, Laura, Podda, Audino, Khan, Rana M. Qasim, Van Damme, Pierre, Kafeja, Froukje and De Coster, Ilse (2011) Safety, immunogenicity and dose ranging of a new Vi-CRM197 conjugate vaccine against typhoid fever: randomized clinical testing in healthy adults. PLoS ONE, 6 (9). e2539. ISSN 1932-6203

Argikar, Upendra, Liang, Guiqing, Bushee, Jennifer, Hosagrahara, Vinayak and Lee, Wendy (2011) Evaluation of pharmaceutical excipients as cosolvents in 4-methyl umbelliferone glucuronidation in human liver microsomes: An application for compounds with low solubility. Drug Metabolism and Pharmacokinetics.

Argikar, Upendra, Mangold, James and Harriman, Shawn (2011) Strategies and Chemical Design Approaches to Reduce the Potential for Formation of Reactive Metabolic Species. Current Topics in Medicinal Chemistry.

Arias, Hugo R, Gu, Ruo-Xu, Feuerbach, Dominik, Guo, Bao-Bao, Ye, Young and Wei, Dong-Qing (2011) Novel Positive Allosteric Modulators of the Human α7 Nicotinic Acetylcholine Receptor. Biochemistry.

Attias-Geva, Zohar, Bentov, Itay, Fishman, Ami, Werner, Haim, Bruchim, Ilan and Jeay, Sebastien (2011) Insulin-like growth factor-I receptor inhibition by specific tyrosine kinase inhibitor NVP-AEW541 in endometroid and serous papillary endometrial cancer cell lines. Gynecologic Oncology. ISSN 0090-8258

B

Baettig, Urs, Akhlaq, Mohammed, Beer, David, Charlton, Steven, Dunstan, Andrew, Bradley, Michelle, Gedeck, Peter, Owen, Charles, Nicklin, Paul, Rosethorne, Elizabeth and Bhalay, Gurdip (2011) Design and synthesis of a library of chemokine antagonists. Bioorganic & Medicinal Chemistry Letters, 21 (21). pp. 6249-6252. ISSN 0960-894X

Baldanzi, Gianluca, Rainero, Elena, Filigheddu, Nicoletta, Mesturini, Riccardo, Song, Shuping, Patrussi, Laura, Zhong, Xiao-Ping, van Blitterswijk, Wim J., Sinigaglia, Fabiola, Nichols, Kim E., Rubio, Ignacio, Pighini, Andrea, Schweighoffer, Tamas, Parolini, Ornella, Graziani, Andrea, Bettio, Valentina, Traini, Sara, Chianale, Federica and Porporato, Paolo E. (2011) SAP-Mediated Inhibition of Diacylglycerol Kinase alpha Regulates TCR-Induced Diacylglycerol Signaling. Journal of Immunology, 187 (11). pp. 5941-5951. ISSN 0022-1767

Baldo, Barbara, Weiss, Andreas, Parker, Christian, Bibel, Miriam, Paganetti, Paolo and Kaupmann, Klemens (2011) A screen for enhancers of clearance identifies huntingtin as an heat shock protein 90 (Hsp90) client protein. Journal of Biological Chemistry, http:/. ISSN 0021-9258

Balibar, Carl, Hollis-Symynkywicz, Micah and Tao, Jianshi (2011) Pantethine Rescues Phosphopantothenoylcysteine Synthetase and Phosphopantothenoylcysteine Decarboxylase Deficiency in Escherichia coli but Not in Pseudomonas aeruginosa. Journal of Bacteriology, 193 (13). pp. 3304-3312. ISSN 0021-9193

Baltus, Christine, Spencer, John, Clegg, William, Press, Neil and Harrington, Ross (2011) Synthesis of a (piperazin-1-ylmethyl)biaryl library via microwave-mediated Suzuki–Miyaura cross-couplings. Tetrahedron Letters, 52 (31). pp. 3963-3968. ISSN 0040-4039

Bassat, Quique, Gonzalez, Raquel, Machevo, Sonia, Nahum, Alain, Lyimo, John, Maiga, Hamma, Martensson, Andreas, Bashraheil, Mahfudh, Ouma, Peter, Ubben, David, Walter, Verena, Nwaiwu, Obiyo, Kipkeu, Chemtai, Lefevre, Gilbert, Ogutu, Bernhards and Menendez, Clara (2011) Similar efficacy and safety of artemether-lumefantrine (Coartem(R)) in African infants and children with uncomplicated falciparum malaria across different body weight ranges. Malaria journal, 10 (1). p. 369. ISSN 1475-2875

Bello, Claudia, Dal Bello, Giovanna, Grossi, Francesco, Patrone, Franco, Ballestrero, Alberto, Dupuis, Marc, Sordat, Bernard, Nencioni, Alessio, Zimmermann, Kaspar, Loretan, Jacqueline, Wartmann, Markus, Vogel, Pierre, Cea, Michele, Motta, Giulia, Moran, Eva, Aubry, Dominique, Nahimara, Aimable, Duchosal, Michel A., Fruscione, Floriana and Pronzato, Paolo (2011) Anti-cancer activity of 5-O-alkyl 1,4-imino-1,4-dideoxyribitols. BIOORGANIC & MEDICINAL CHEMISTRY, 19 (24). pp. 7720-7727. ISSN 0968-0896

Benoit, Roger and Auer, Manfred (2011) A direct way of redox sensing. RNAbiology, 8 (1). pp. 1-6. ISSN 1547-6286

Bielen, Aleksandra, Perryman, Lara, Box, Gary, Valenti, Melanie, de Haven Brandon, Alexis, Martins, Vanessa, Jury, Alexa, Popov, Sergey, Jeay, Sebastien, Raynaud, Florence, Hofmann, Francesco, Hargrave, Darren, Eccles, Sue and Jones, Chris (2011) Enhanced efficacy of IGF1R inhibition in paediatric glioblastoma by combinatorial targeting of PDGFRa/b. Molecular Cancer Therapeutics, 10 (8). pp. 1407-1418. ISSN 1535-7163

Bifani, Juan Pablo, Lefèvre, Philippe, Wang, Xiao-Ming, Karine, Soetaert, Rens, Céline, De Bruyn, Jacqueline, Lanéelle, Marie-Antoinette, Houyoux, Nicolas, Laval, Françoise, Lemassu, Anne, Wattiez, Ruddy, Daffé, Mamadou and Fontaine, Véronique (2011) Cpn60.1/GroEL-1/Hsp60-1, a New Potential Antimycobacterial Drug Target Involved in Antibiotics Resistance. Microbiology, 157 (4). pp. 1205-1219. ISSN 1608-3237; 0026-2617

Block, Stan L, Yogev, Ram, Waldmeier, Felix and Hamed, Kamal (2011) Safety and pharmacokinetics of a single 1500-mg dose of famciclovir in adolescents with recurrent herpes labialis. The Pediatric infectious disease journal, 30 (6). pp. 525-528. ISSN 1532-0987

Bonavia, Aurelio, Franti, Michael, Keaney, Erin, Kuhen, Kelli, Seepersaud, Mohindra, Radetich, Branko, Shao, Jian, Honda, Ayako, Dewhurst, Janetta, Balabanis, Kara, Monroe, James, Wolff, Karen, Osborne, Colin, Bourque, Leanne, Hoffmaster, Keith, Amin, Jakal, Markovits, Judit, Broome, Michelle, Skuba, Elizabeth, Cornella-Taracido, Ivan, Joberty, Gerard, Bouwmeester, Antonius, Hamann, Lawrence, Tallarico, John, Tommasi, Ruben, Compton, Teresa and Bushell, Simon (2011) Identification of Pyrimidine Biosynthesis Inhibitors with Broad Spectrum Antiviral Activity and Assessment of the Druggability of this Pathway for Efficacy against RSV. Proceedings of the National Accademy of Sciences USA, 108 (17). pp. 6739-6744. ISSN 0027-8424

Bornancin, Frederic (2011) Ceramide kinase: The first decade. Cellular Signalling, 23 (6). pp. 999-1008. ISSN 0898-6568

Boulton, Craig, Meiser, Karin, David, Olivier J and Schmouder, Robert (2011) Pharmacodynamic Effects of Steady-State Fingolimod on Antibody Response in Healthy Volunteers: A 4-Week, Randomized, Placebo-Controlled, Parallel-Group, Multiple-Dose Study. Journal of clinical pharmacology. ISSN 0091-2700

Brennan, Orlaith, Kennedy, OD, Lee, TC, Rackard, SM, O'Brien, FJ, McNamara, LM and Gasser, Juerg Andreas (2011) The Effects of Estrogen Deficiency and Bisphosphonate Treatment on Tissue Mineralisation and Stiffness in an Ovine Model of Osteoporosis. Journal of Biomechanics or Bone, 44 (3). pp. 386-390. ISSN 0021-9290

Brocklehurst, Cara, Laumen, Kurt, La Vecchia, Luigi, Shaw, Duncan and Voegtle, Markus (2011) Diasteroisomeric Salt Formation and Enzyme-Catalyzed Kinetic Resolution as Complimentary Methods for the Chiral Separation of cis/trans-Enantiomers of 3-Aminocyclohexanol. Organic Process Research and Development, 15 (1). pp. 294-300. ISSN 1083-6160

Brocklehurst, Cara, Lehmann, Hansjoerg and La Vecchia, Luigi (2011) Nitration Chemistry in Continuous Flow using Fuming Nitric acid in a Commercially Available Flow Reactor. Organic Process Research and Development. ISSN 1083-6160

Burger, Matthew, Pecchi, Sabina, Wagman, Allan, Ni, Zhijie, Knapp, Mark, Hendrickson, Thomas, Atallah, Gordana, Pfister, Keith, Zhang, Yanchen, Bartulis, Sarah, Ng, Simon, Verhagen, Joelle, Huh, Kay, Iwanowicz, Edwin, Menezes, Daniel, Merritt, Hanne, Lee, Isabelle, Weismann, Marion, Kaufman, Susan, Crawford, Kenneth, Chin, Michael, Bussiere, Dirksen, Shoemaker, Kevin, Verhagen, Joelle, Frazier, Kelly, Xin, Xiaohua, Haznedar, Joshua, Zaror, Isabel, Maira, Sauveur-Michel and Voliva, Charles (2011) Identification of NVP-BKM120 as a Potent, Selective, Orally Bioavailable Class I PI3 Kinase Inhibitor for Treating Cancer. ACS Medicinal Chemistry Letters, 2 (10). pp. 774-779. ISSN 1948-5875

Burton, Victoria, Holmes, Alan, Ciuclan, Loredana, Robinson, Alexander, Roger, Jan, Jarai, Gabor, Pearce, Andrew and Budd, David (2011) Attenuation of leukocyte recruitment via inhibition of CXCR1/2 inhibition stops the progression of PAH in mice with genetic ablation of endothelial BMPR-II. Blood, 118 (17). pp. 4750-4758. ISSN 0006-4971

Bushee, Jennifer and Argikar, Upendra (2011) An experimental approach to enhance parent ion fragmentation for metabolite identification studies: Application of dual collision cells in an orbital trap. Rapid Communications in Mass Spectrometry, 25 (10). pp. 1356-1362. ISSN 1097-0231

beeh, kai, wagner, frank, Khindri, Sanjeev and Drollmann, Anton Franz (2011) Effect of indacaterol on dynamic lung hyperinflation and breathlessness in patients with COPD. COPD, 8 (5). pp. 340-345. ISSN 1541-2555

C

Cao, Xueying, Erdemli, Gul, Urban, Laszlo, Lee, Yan, Golden, Andrew, Holmqvist, Mats, Li, Nianzhen, Chen, Quin, Nevill, Tanner, Johnson, Juliette and Ionescu-Zanetti, Christian (2011) IonFlux, a Microfluidic Patch Clamp System Evaluated with hERG Channel Physiology and Pharmacology. Assay and Drug Development Technologies.

Cao, Yiqun and Landrum, Gregory (2011) Inchi wrappers for the RDKit. RDKit: open source cheminformatics.

Carcache, David, Vranesic, Ivan-Toma, Blanz, Joachim, Desrayaud, Sandrine, Fendt, Markus and Glatthar, Ralf (2011) Benzimidazoles as potent and orally active mGlu5 receptor antagonists with an improved PK profile. ACS Medicinal Chemistry Letters, 2 (1). pp. 58-62. ISSN 1948-5875

Caughlan, Ruth, Jones, Adriana, Delucia, Angela, Woods, Angela, Xie, Lili, Ma, Bing, Barnes, Whitney, Walker, John, Sprague, Elizabeth, Yang, Xia and Dean, Charles (2011) Mechanisms decreasing in vitro susceptibility to the LpxC inhibitor CHIR-090 in the Gram negative pathogen Pseudomonas aeruginosa. Antimicrobial Agents and Chemotherapy. ISSN 0066-4804

Chapelat, Julien, Berst, Frederic, Marzinzik, Andreas, Moebitz, Henrik, Drueckes, Peter, Fabbro, Doriano, Trappe, Joerg and Seebach, Dieter (2011) Substrate profiling of IGF-1R and InsR: Identification of a potent pentamer substrate. Bioorganic and Medicinal Chemistry Letters.

Chen, Jian, Shen, Qiong, Labow, Mark and Gaither, L Alex (2011) Protein kinase D3 sensitizes RAF inhibitor RAF265 in melanoma cells by preventing reactivation of MAPK signaling. Cancer research, 71 (12). pp. 4280-4291. ISSN 1538-7445

Chen, Xiao-Hui, Zhao, Hongjuan, Hatsis, Panagiotis and Amin, Jakal (2011) Investigation of Dried Blood Spot Card-Induced Interferences in Liquid Chromatography/Mass Spectrometry. Journal of Pharmaceutical and Biomedical Analysis. ISSN 0731-7085

Chiong, Edmund, Lee, I-Ling, Dadbin, Ali, Sabichi, Anita L, Harris, Loleta, Urbauer, Diana, McConkey, David, Grossman, H Barton and Imark, Esther (2011) Effects of mTOR Inhibitor Everolimus (RAD0011) On Bladder Cancer Cells. Clinical Cancer Research, 17 (9). pp. 2863-2873. ISSN 1078-0432

Christen, Selina, Holdener, Martin, Beerli, Christian, Thoma, Gebhard, Bayer, Monika, Pfeilschifter, Josef, Hintermann, Edith, Zerwes, Hans-Guenter and Christen, Urs (2011) Small molecule CXCR3 antagonist NIBR2130 has only a limited impact on type 1 diabetes in a virus-induced mouse model. Clinical and experimental immunology, 165 (3). pp. 318-328. ISSN 0009-9104

Ciuclan, Loredana, Bonneau, Olivier, Hussey, Martin, Duggan, Nicholas, Holmes, Alan, Good, Robert, Stringer, Rowan, Jones, Peter, Morrell, Nicholas W., Jarai, Gabor, Walker, Christoph, Westwick, John and Thomas, Matthew (2011) A Novel Murine Model of Severe Pulmonary Arterial Hypertension. American Journal of Respiratory and Critical Care Medicine. ISSN 1073-449X

Coan, Kristin, Ottl, Johannes and Klumpp, Martin (2011) Non-stoichiometric Inhibition in High-Throughput Screening. Expert Opinion on Drug Discovery.

Collingwood, Steve, Ratcliffe, Andrew and Allen, Jack (2011) Kinase Inhibitors from Early Research to Clinic. Drugs of the Future, 36 (3). pp. 249-263. ISSN 0377-8282

Commerford, Susan, He, Xiaohui, Liu, Hong, Seidel, Martin, Jaton, Anne-Lise, Gromada, Jesper, Teixeira, Sandra, Gerber, Sarah, Chen, Alice, Dardik, Beatriz, Chaperon, Frederique, Schwartzkopf, Chad, Nguyen-Tran, Van, Hollenbeck, Thomas and Mcnamara, Peter (2011) Characterization of a novel, brain-penetrating CB1 receptor inverse agonist: metabolic profile in diet-induced obese models and aspects of central activity. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 384 (6). pp. 565-581. ISSN 0028-1298

Connolly, Michael K., Ayo, Diego, Hackman, Michael, Malhotra, Ashim, Bedrosian, Andrea S., Ibrahim, Junaid, Cieza-Rubio, Napoleon E., Nguyen, Andrew H., Henning, Justin R., Pachter, H. Leon and Miller, George (2011) Dendritic Cell Depletion Exacerbates Acetaminophen Hepatotoxicity. Hepat0logy, 54 (3). pp. 959-968. ISSN 0270-9139

Cottens, Sylvain and Cottens, Sylvain (2011) Perspective on Future Medicinal Chemistry. Futurescience, 3 (15). pp. 1863-1872. ISSN 1759-6180

Craig, Ian (2011) PocketAnalyzerPCA. Project is software (source code) to be "published" as download from a website.

Craig, Ian, Pfleger, Christopher, Gohlke, Holger, Essex, Jonathan and Spiegel, Katrin (2011) Pocket-space maps to identify novel binding-site conformations in proteins. Journal of Chemical Information and Modeling.

Curtis, Allison, Calabro, Katherine, Galarneau, Jean-Rene, Bigio, Irving and Krucker, Thomas (2011) Temporal Variations in Skin Pigmentation of C57Bl/6 Mice Affect Optical Bioluminescence Quantitation. Molecular Imaging and Biology, 13 (6). pp. 1114-1123. ISSN 1536-1632

D

Dalvit, Claudio and Vulpetti, Anna (2011) Fluorine-Protein Interactions and 19F NMR Isotropic Chemical Shift: An Empirical Correlation. ChemMedChem, 6 (1). pp. 104-114. ISSN 1860-7179

Delucia, Angela, Six, David, Caughlan, Ruth, Gee, Patricia, Hunt, Ian, Lam, Joseph and Dean, Charles (2011) Lipopolysaccharide inner-core phosphates are required for complete LPS synthesis and transport to the outer membrane in Pseudomonas aeruginosa PAO1. mBio, 2 (4). pii: e00142. ISSN 2150-7511

Deng, Gejing, Lee, Lac, Chenail, Gregg, Palestrant, Deborah, Whitehead, Lewis, Sachdeva, Meena, Dzink-Fox, Joann, Lamarche, Matthew and Leeds, Jennifer (2011) In vitro and in vivo activities of novel, semisynthetic thiopeptide inhibitors of bacterial elongation factor Tu. Antimicrobial Agents and Chemotherapy, 55 (11). pp. 5277-5283. ISSN 0066-4804

Deng, Gejing, Lee, Lac, Chenail, Gregg, Palestrant, Deborah, Whitehead, Lewis, Sachdeva, Meena, Lamarche, Matthew and Leeds, Jennifer (2011) In vitro and in vivo activities of novel, semisynthetic thiopeptide inhibitors of bacterial elongation factor Tu. Antimicrobial Agents and Chemotherapy, 55 (11). pp. 5277-5283. ISSN 0066-4804

Dertinger, Stephen D., Phonethepswath, Souk, Weller, Pamela, Nicolette, John, Murray, Joel, Sonders, Paul, Vohr, Hans-Werner, Shi, Jing, Krsmanovic, Ljubica, Gleason, Carol, Custer, Laura, Henwood, Andrew, Sweder, Kevin, Stankowski Jr, Leon F., Roberts, Daniel J., Giddings, Amanda, Kenny, Julia, Lynch, Anthony M., Defrain, Céline, Nesslany, Fabrice, van der Leede, Bas-jan M., Van Doninck, Terry, Schuermans, Ann, Tanaka, Kentaro, Hiwata, Yoshie, Tajima, Osamu, Eleanor, Wilde, Elhajouji, Azeddine, Gunther, William C., Thiffeault, Catherine J., Shutsky, Thomas J., Fiedler, Ronald D., Kimoto, Takafumi, Bhalli, Javed A., Heflich, Robert H. and MacGregor, James T. (2011) International Pig-a gene mutation assay trial: Evaluation of transferability across fourteen laboratories. Environmental and Molecular Mutagenesis, 52 (9). pp. 690-698. ISSN 0893-6692

Deschwanden, Alexandra, Karolewicz, Beata, Feyissa, Anteneh, M, Treyer, Valerie, Ametamey, Simon, M, Johayem, Annas, Burger, Cyrill, Auberson, Yves, Sovago, Judit, Stockmeier, Craig, A, Buck, Alfred and Hasler, Gregor (2011) Reduced Metabotropic Glutamate Receptor 5 Density in Major Depression Determined by [11C]ABP688 Positron Emission Tomography and Postmortem Study. American Journal of Psychiatry, 168 (7). pp. 727-734. ISSN 0002-953X

Didiot, Marie-Cecile, Serafini, Sergio, Pfeifer, Martin, King, Frederick and Parker, Christian (2011) Multiplexed Reporter Gene Assays: Monitoring the cell viability and the compound kinetics on luciferase activity. Journal of Biomolecular Screening, 16 (7). pp. 786-793. ISSN 1087-0571

Djimdé, Abdoulaye A, Tekete, Mamadou, Abdulla, Salim, Lyimo, John, Bassat, Quique, Mandomando, Inacio, Lefèvre, Gilbert and Borrmann, Steffen (2011) Pharmacokinetic and pharmacodynamic characteristics of a new pediatric formulation of artemether-lumefantrine in African children with uncomplicated Plasmodium falciparum malaria. Antimicrobial agents and chemotherapy, 55 (9). pp. 3994-3999. ISSN 1098-6596

Doghman, Mabrouka, Axelson, Magnus and Lalli, Enzo (2011) Potent inhibitory effect of the cyclolignan picropodophyllin (PPP) on human adrenocortical carcinoma cells proliferation. American journal of cancer research, 1 (3). pp. 356-361. ISSN 2156-6976

Drollmann, Anton Franz, Crane, Helen, Di Scala, Lilla and Fogarty, Charles (2011) Bronchodilatory effects of NVA237, a once daily long-acting muscarinic antagonist, in COPD patients. Respiratory Medicine, 105 (3). pp. 337-342. ISSN 0954-6111

Duttaroy, Alokesh, Voelker, Frank, Merriam, Kimberly, Zhang, Xia, Ren, Xianglin, Subramanian, Kala, Hughes, Thomas and Burkey, Bryan (2011) The DPP-4 Inhibitor Vildagliptin Increases Pancreatic Beta Cell Mass In Neonatal Rats. European Journal of Pharmacology, 650 (2-3). pp. 703-707. ISSN 0014-2999

de backer, jan, de backer, wilhelm, vos, w. g., vinchurkar, s., claes, r., wulfrank, p., parizel, p., germonpre, p. and Drollmann, Anton Franz (2011) Validation of computational fluid dynamics in CT-based airway models with SPECT/CT. Radiology, 257 (3). pp. 854-862. ISSN 0033-8419

E

Emotte, Corinne, Deglave, Fanny, Heudi, Olivier, Picard, Franck and Kretz, Olivier (2011) Fast simultaneous quantitative analysis of FTY720 and its metabolite FTY720-P in human blood by on-line solid phase extraction coupled with tandem liquid chromatography mass spectrometry. Journal of Pharmaceutical and biomedical analysis, 58. pp. 102-112. ISSN 0731-7085

Ettenger, R, Schmouder, R, Kovarik, J M, Bastien, M C and Hoyer, P F (2011) Pharmacokinetics, pharmacodynamics, safety, and tolerability of single-dose fingolimod (FTY720) in adolescents with stable renal transplants. Pediatric transplantation, 15 (4). pp. 406-413. ISSN 1399-3046

Eucker, Tyson P. and Konkel, Michael E. (2011) The cooperative action of bacterial fibronectin-binding proteins and secreted proteins promote maximal Campylobacter jejuni invasion of host cells by stimulating membrane ruffling. Cellular Microbiology. ISSN 1462-5814

F

Faller, Bernard, Berellini, Giuliano, Ertl, Peter, Ottaviani, Giorgio and Collis, Alan (2011) Can History Foretell Future ? Drug Discovery Today, 16 (21-22). pp. 976-984. ISSN 1359-6446

Ferrand, Sandrine, Tao, Jianshi, Shen, Xiaoyu, Mcguire, Dorothy, Schmid, Andres, Glickman, Fraser and Schopfer, Ulrich (2011) Screening for Mevalonate Pathway Inhibitors using sensitized bacteria strains. Journal of Biomolecular Screening, 16 (6). pp. 637-646. ISSN 1087-0571

Ferreira, I.L., Bajouco, L.M., Oliveira, C.R., Auberson, Yves, Rego, A.C. and Mota, S.I. (2011) Amyloid beta peptide 1-42 disturbs intracellular calcium homeostasis through activation of GluN2B-containing N-methyl-D-aspartate receptors in cortical cultures. Cell Calcium. ISSN 0143-4160

Fetar, Hossam, Christie, Gilmour, Rachel, Klinoski, Daigle, Denis, Dean, Charles and Poole, Keith (2011) The mexEF-oprN multidrug efflux operon of P. aeruginosa: regulation by the MexT activator in response to nitrosative stress and chloramphenicol. Antimicrobial Agents and Chemotherapy, 55 (2). pp. 508-514. ISSN 0066-4804

Fiorina, Paolo, Pietramaggiori, Giorgio, Scherer, Saja, Jurewicz, Mollie, Mathews, Jasmine, Vergani, Andrea, Thoma, Gebhard, Orsenigo, Elena, Staudacher, Carlo, La Rosa, Stefano, Capella, Carlo, Carothers, Adelaide, Zerwes, Hans-Guenter, Luzi, Livio, Abdi, Reza and Orgill, Dennis (2011) The mobilization and effect of endogenous bone marrow progenitor cells in diabetic wound healing. Cell Transplantation, 19 (11). pp. 1369-1386. ISSN 0963-6897

Fonseca, Sonya, Gromada, Jesper and Urano, Fumihiko (2011) ER stress: The link between pancreatic beta cell dysfuntion and death. Trends in Endocrinology and Metabolism.

Fonseca, Sonya, Urano, Fumihiko, Burcin, Mark and Gromada, Jesper (2011) Stress HypERactivation in the Beta Cell. Islets, 2 (1). pp. 1-9. ISSN 1938-2014

Forbes, Ben, Asgharian, Bahman, Dailey, Lea Ann, Ferguson, Douglas, Gerde, Per, Gumbleton, Mark, Gustavsson, Lena, Hardy, Colin, Hassall, David, Jones, Rhys, Lock, Ruth, Maas, Janet, McGovern, Tim, Pitcairn, Gary R, Somers, Graham and Wolff, Ron K (2011) Challenges in inhaled product development and opportunities for open innovation. Advanced drug delivery reviews, 63 (1-2). pp. 69-87. ISSN 1872-8294

Freeman, Mark, Hardaker, Liz, Banner, Kathy, Poll, Christopher, Coulthard, Alex and Dewhurst, Jennifer (2011) Effects of a combination of subchronic tobacco smoke exposure and lipopolysaccharide administration on pulmonary inflammation in the mouse. British Journal of Pharmacology, 8 (1). 132P.

Fu, Qiang, Berbee, Maaike, Wang, Wenze, Boerma, Marjan, Schmid, Herbert and Hauer-Jensen, Martin (2011) Preclinical evaluation of SOM230 as a radiation mitigator in a mouse model: post-exposure time window and mechanisms of action. Radiation Research, 175 (6). pp. 728-735. ISSN 0033-7587

Fu, Yunlin, Li, Wenkui, Smith, Harold and Tse, Francis (2011) A practical approach to address the issue of analyte nonspecific binding in quantitative analysis of untreated and transferred urine samples. Bioanalysis, 3 (9). pp. 967-972. ISSN 1757-6180

G

Garofalo, Cecilia, Manara, Maria Christina, Nicoletti, Giordano, Marino, Maria Theresa, Nanni, Patrizia, Lollini, Pier-Luigi, Prandini, Giuseppe, Lopez-Guerrero, José Antonio, Schaefer, Karl-Ludwig, Belfiore, Antonino, Picci, Piero and Scotlandi, Katia (2011) Efficacy of and resistance to anti‐IGF‐1R therapies in sarcomas is dependent on Insulin Receptor signaling. Oncogene, 30 (24). pp. 2730-2740. ISSN 0950-9232

Garofolo, Fabio, Rocci Jr., Mario, Dumont, Isabelle, Martinez, Suzanne, Lowes, Steve, Woolf, Eric, van Amsterdam, Peter, Bansal, Surendra, Gomes Barra, Airadna, Bauer, Ronald, Booth, Brian, Carrasco-Triguero, Montserrat, DeSilva, Binodh, Dunn, John, Gallicano, Keith, Gouty, Dominique, Ho, Stacy, Hucker, Richard, Jemal, Mohammed, Katori, Noriko, Le Blaye, Olivier, Lee, Jean, Li, Wenkui, Michael, Steve, Nehls, Corey, Nicholson, Robert, Ormsby, Eric, Tang, Daniel, Viswanathan, C, Wiener, Russel and Young, Graeme (2011) 2011 White Paper on Recent Issues in Bioanalysis & Regulatory Findings from Audits and Inspections. Bioanalysis, 3 (18). pp. 2081-2096. ISSN 1757-6180

Giovannoni, Jerome and Peltier, John (2011) Implementation of high-throughput quality control processes within Compound Management. European Pharmaceutical Review, 16 (4). pp. 49-52.

Glick, Meir and Jacoby, Edgar (2011) The Role of Computational Methods in the Identification of Bioactive Compounds. Current Opinion in Chemical Biology. ISSN 1367-5931

Glowienke, Susanne (2011) Practical experience of in silico assessment for genotoxic impurities. Regul Pharm Tox.

Gomez-Mancilla, Baltazar (2011) Challenges and opportunities of criteria alignment regarding Neurodegenerative Diseases. World Health Summit.

Gossert, Alvar, Hinniger, Alexandra, Gutmann, Sascha, Jahnke, Wolfgang, Strauss, Andre and Fernandez, Cesar (2011) A simple protocol for amino acid type selective isotope labeling in insect cells with improved yields and high reproducibility. Journal of Biomolecular NMR.

Gottar-Guillier, Marie, Dodeller, Francis, Huesken, Dieter, Iourgenko, Vadim, Mickanin, Craig, Labow, Mark, Kinzel, Bernd, Mueller, Matthias, Gaveriaux, Samuel, Alitalo, Kari, Littlewood-Evans, Amanda and Cenni, Bruno (2011) The tyrosine kinase BMX is an essential mediator of inflammatory arthritis in a kinase-independent manner. Journal of Immunology, 186 (10). pp. 6014-6023. ISSN 0022-1767

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Saul, Allan (2011) Vaccines for Neglected Diseases. In: Vaccine Design: Innovative Approaches and Novel Strategies. Caister Academic Press, pp. 243-252. ISBN 978-1-904455-74-5

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