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Blank, Jutta, Hintermann, Samuel, Schneider, Nadine, Schuffenhauer, Ansgar and Shultz, Michael (2020) Outline for a Perspective Article on Novartis’ approach to compound screening for hit and lead finding and the design of compounds sets for diversity driven screening. Journal of medicinal chemistry for publisher only.

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Chen, Hui, Sun, Shuhao, Liu, Yahu and Liao, Xuebin (2020) Nickel-Catalyzed Cyanation of Aryl Halides and Hydrocyanation of Alkynes via C-CN Bond Cleavage and Cyano Transfer. ACS Catalysis, 10. pp. 1397-1405. ISSN 2155-54352155-5435

Chianelli, Donatella, Rucker, Paul, Tully, David, Nelson, John, Liu, Xiaodong, Bursulaya, Badry, Hernandez, Eloy , Chu, Alan, Schmeits, James, Hill, Robert, Bao, Dingjiu, Zoll, Jocelyn, Kim, Young, Groessl, Todd, McNamara, Peter, Richmond, Wendy, Sancho Martinez, Ignacio, Badman, Michael, Molteni, Valentina, Jason, Roland, Jane, Wu, David, Huang, Bo, Liu, Andrew, Phimister, Martin, Seidel, Sean, Joseph, Bryan, Laffitte, Prashad, Mahavir, Schlama, Thierry and Liu, Yugang (2020) Nidufexor (LMB763), a Novel FXR Modulator for the Treatment of Nonalcoholic Steatohepatitis. Journal of medicinal chemistry, 63 (8). pp. 3868-3880. ISSN 9b01621

Chianelli, Donatella, Rucker, Paul, Tully, David, Nelson, John, Liu, Xiaodong, Bursulaya, Badry, Hernandez, Eloy , Chu, Alan, Schmeits, James, Hill, Robert, Bao, Dingjiu, Zoll, Jocelyn, Kim, Young, Groessl, Todd, McNamara, Peter, Richmond, Wendy, Sancho Martinez, Ignacio, Badman, Michael, Molteni, Valentina, Jason, Roland, Jane, Wu, David, Huang, Bo, Liu, Andrew, Phimister, Martin, Seidel, Sean, Joseph and Bryan, Laffitte (2020) Nidufexor (LMB763), a Novel FXR Modulator for the Treatment of Nonalcoholic Steatohepatitis (NASH). Journal of medicinal chemistry, 63 (8). pp. 3868-3880. ISSN 9b01621

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Grande, Enrique, Giovannini, Monica, Marriere, Eddie, Pultar, Philippe, Quinlan, Michelle, Chen, Heller, Curigliano, Giuseppe and Cui, Xiaoming (2020) Effect of capmatinib on the pharmacokinetics of digoxin and rosuvastatin administered as a two-drug cocktail in patients with MET-dysregulated advanced solid tumors: A phase I, multicenter, open-label, single-sequence drug-drug interaction study. British Journal of Clinical Pharmacology.

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Huppertz, Christine, Wieczorek, Grazyna, Littlewood-Evans, Amanda, Oliver, Stephen, Jaeger, Benedikt, Engelhard, Peggy, Bauernfeind, Franz-Georg, Welte, Tobias, Hornung, Veit and Prasse, Antje (2020) The NLRP3 inflammasome pathway is activated in sarcoidosis and involved in granuloma formation. The European respiratory journal. ISSN 13993003

Isalomboto Nkanga, Christian , Fisch, Andreas, Rad-Malekshahi, Mazda , Duvnjak Romic, Marieta, Kittel, Birgit, Ullrich, Thomas, Wang, Jing, Werner Maçedo Krause, Rui, Adler, Sabine, Lammers, Twan, Hennink, Wim and Ramazani, Farshad (2020) Clinically established biodegradable long acting injectables: An industry perspective. Advanced drug delivery reviews, 167. pp. 19-46. ISSN 33202261

Isobe, Yosuke, Okumura, Mikiko, McGregor, Lynn, Brittain, Scott, Jones, Michael, Liang, Xiaoyou, White, Ross, Forrester, William, McKenna, Jeffrey, Tallarico, John, Schirle, Markus, Maimone, Thomas and Nomura, Daniel (2020) Manumycin polyketides act as molecular glues between UBR7 and P53. Nature chemical biology. ISSN 1552-4469; 1552-4450

Jahnke, Wolfgang, Erlanson, Daniel A, de Esch, Iwan JP, Johnson, Christopher N, Mortenson, Paul N, Ochi, Yuji and Urushima, Tatsuya (2020) Fragment-to-Lead Medicinal Chemistry Publications in 2019. Journal of Medicinal Chemistry, 63 (24). pp. 15494-15507. ISSN 15204804

James, Alexander David, Schiller, Hilmar, Marvalin, Cyrille, Jin, Yi, Borell, Hubert, Roffel, Ad , Glaenzel, Ulrike, Ji, Yan and Camenisch, Gian P. (2020) An integrated assessment of the ADME properties of the CDK4/6 Inhibitor ribociclib utilizing preclinical in vitro, in vivo and human ADME data. Pharmacology Research & Perspectives, 8 (3). ISSN 2052-17072052-1707

Jayawardena, Asitha, Liu, Tingyu, Pereira, Bernard, Wang, Ye, Baker, Lisa, Leary, Rebecca, Sabatos-Peyton, Catherine and Hartnick, Christopher (2020) Genetic variation in twins with vastly different phenotypical expression of recurrent respiratory papillomatosis. The Laryngoscope. ISSN 1531-4995

Jentsch, Marcel, Snyder, Petra, Sheng, Caibin, Cristiano, Elena and Loewer, Alexander (2020) p53 dynamics in single cells are temperature-sensitive. Scientific reports, 10 (1). p. 1481. ISSN 2045-2322

Ji, Yan, Abozeid, Ahmed M, Samant, Tanay, Yang, Shu and Rodriguez Lorenc, Cristina (2020) Evaluation of Absolute Oral Bioavailability and Bioequivalence of Ribociclib, a Cyclin-Dependent Kinase 4/6 Inhibitor, in Healthy Subjects. Clinical Pharmacology in Drug Development. ISSN 21607648

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Johnson, Erik C. B., Ho, Kaitlyn, Das, Melanie, Sanchez , Pascal, Djukic, Biljana, Yu, Xinxing, Lopez, Isabel, Gill, Michael, Paz, Jeanne, Palop, Jorge and Mucke, Lennart (2020) Behavioral and neural network abnormalities of human APP transgenic mice resemble those of App knockin mice but are not prevented by early inhibition of BACE1. Molecular neurodegeneration, 15 (1).

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Jones, Graham, Chirino Chace, Bernardita and Wright, Justin (2020) Cultural diversity drives innovation: empowering teams for success. International Journal of Innovation Science, 12 (3). pp. 323-343. ISSN 1757-2223

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Junker Walker, Ursula (2020) Histological thymus alterations in rats treated with a S1P receptor agonist. European society of toxicologic pathology website: "Guess what" the diagnotic cases of the ESTP.

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Kaul, Martin, Jarvis, Philip, Rozenberg, Izabela, Kolbinger, Frank, Di Padova, Franco E., Calonder, Claudio, Espie, Pascal, Rondeau, Jean-Michel, Cebe, Regis, Huber, Thomas, Mussmann, Rainer and Aassi, Maher (2020) First-in-human study demonstrating the safety and clinical efficacy of novel anti-IL-17A monoclonal antibody CJM112 in moderate to severe plaque psoriasis. Journal of the European Academy of Dermatology and Venereology, 2020 (4). pp. 1-9. ISSN 14683083

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